ARRAY BIOPHARMA, INC.
Patent Owner
Stats
- 184 US PATENTS IN FORCE
- 11 US APPLICATIONS PENDING
- Feb 27, 2018 most recent publication
Details
- 184 Issued Patents
- 0 Issued in last 3 years
- 0 Published in last 3 years
- 5,329 Total Citation Count
- Oct 27, 1998 Earliest Filing
- 89 Expired/Abandoned/Withdrawn Patents
Patent Activity in the Last 10 Years
Technologies
Intl Class
Technology
Matters
Rank in Class
Top Patents (by citation)
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Recent Publications
Publication #
Title
Filing Date
Pub Date
Intl Class
2017/0260,589 POINT MUTATIONS IN TRK INHIBITOR-RESISTANT CANCER AND METHODS RELATING TO THE SAMEOct 26, 16Sep 14, 17[A61K, C12Q]
2017/0252,317 N4-PHENYL-QUINAZOLINE-4-AMINE DERIVATIVES AND RELATED COMPOUNDS AS ERBB TYPE I RECEPTOR TYROSINE KINASE INHIBITORS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASESMay 19, 17Sep 07, 17[A61K, C07D]
2017/0096,425 SUBSTITUTED PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS RET KINASE INHIBITORSJul 15, 16Apr 06, 17[A61K, C07D]
2017/0087,156 1-((3S,4R)-4-(3-FLUOROPHENYL)-1-(2-METHOXYETHYL)PYRROLIDIN-3-YL)-3-(4-METHYL-3-(2-METHYLPYRIMIDIN-5-YL)-1-PHENYL-1H-PYRAZOL-5-YL)UREA AS A TRKA KINASE INHIBITORMay 14, 15Mar 30, 17[A61K, C07D]
Recent Patents
Patent #
Title
Filing Date
Issue Date
Intl Class
9896435 N-pyrrolidinyl,N′-pyrazolyl-urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitorsNov 12, 13Feb 20, 18[C07D]
9889134 Polymorphs of ARRY-380, a selective HER 2 inhibitor and pharmaceutical compositions containing themOct 26, 15Feb 13, 18[A61K, C07D, A61P]
9878997 Pyrrolidinyl urea, pyrrolidinyl thiourea and pyrrolidinyl guanidine compounds as TrkA kinase inhibitorsDec 16, 16Jan 30, 18[C07D]
9828360 Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitorsNov 13, 13Nov 28, 17[C07D]
9822118 Bicyclic heteroaryl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitorsNov 13, 13Nov 21, 17[C07D]
9809578 Pyrazolyl urea, thiourea, guanidine and cyanoguanidine compounds as trkA kinase inhibitorsNov 13, 13Nov 07, 17[C07D]
Expired/Abandoned/Withdrawn Patents
Patent #
Title
Status
Filing Date
Issue/Pub Date
Intl Class
2016/0251,350 CRYSTALLINE FORMS OF A PYRROLOPYRIDINE COMPOUNDAbandonedFeb 26, 16Sep 01, 16[A61K, C07D]
2016/0235,754 HYDROXYLATED AND METHOXYLATED PYRIMIDYL CYCLOPENTANES AS AKT PROTEIN KINASE INHIBITORSAbandonedApr 28, 16Aug 18, 16[A61K]
2016/0137,608 SUBSTITUTED BENZOAZEPINES AS TOLL-LIKE RECEPTOR MODULATORSAbandonedOct 13, 15May 19, 16[C07D]
2016/0137,654 CRYSTALLINE FORM OF (S)-N-(5-((R)-2-(2,5-DIFLUOROPHENYL)-PYRROLIDIN-1-YL)-PYRAZOLO[1,5-A]PYRIMIDIN-3-YL)-3-HYDROXYPYRROLIDINE-1-CARBOXAMIDE HYDROGEN SULFATEAbandonedNov 16, 15May 19, 16[C07D]
2015/0299,182 CRYSTALLINE FORMS OF (1S)-1-[5-(AMINO)-1,2,4-THIADIAZOL-3-YL]ETHANE-1,2-DIOLAbandonedNov 08, 13Oct 22, 15[C07D]
2015/0231,117 ARRY-520 FOR USE IN TREATING CANCER IN A PATIENT WITH LOW AAGAbandonedAug 13, 13Aug 20, 15[A61K, G01N]
2015/0191,479 DIHYDROFURO PYRIMIDINES AS AKT PROTEIN KINASE INHIBITORSAbandonedOct 16, 14Jul 09, 15[A61K, C07D]
2015/0045,391 FILANESIB COMBINED WITH POMALIDOMIDE DISPLAYS ENHANCED ANTI-TUMOR ACTIVITYAbandonedAug 07, 14Feb 12, 15[A61K]
2014/0315,887 PYRIMIDYL CYCLOPENTANES AS AKT PROTEIN KINASE INHIBITORSAbandonedJul 01, 14Oct 23, 14[C07D]
2014/0309,226 PIPERIDINYL-SUBSTITUTED CYCLIC UREAS AS GPR119 MODULATORSAbandonedNov 14, 12Oct 16, 14[C07D]
2014/0256,756 PIPERIDINYL-SUBSTITUTED LACTAMS AS GPR119 MODULATORSAbandonedOct 30, 12Sep 11, 14[C07D]
2014/0018,399 MITOTIC KINESIN INHIBTORS AND METHODS OF USE THEREOFAbandonedSep 19, 13Jan 16, 14[C07D]
2013/0184,257 PIPERIDINYL-SUBSTITUTED LACTAMS AS GPR119 MODULATORSAbandonedSep 15, 11Jul 18, 13[C07D]
2013/0065,908 DIHYDROFURO PYRIMIDINES AS AKT PROTEIN KINASE INHIBITORSAbandonedNov 08, 12Mar 14, 13[A61K, C07D, A61P]
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